I-Pure Rotundine Powder(l-tetrahydropalmatine,l-THP)

Amanye Amagama:I-L-Tetrahydropalmatine
Umthombo Wezitshalo:Stephania tetrandra or Corydalis yanhusuo
Inombolo ye-CAS:10097-84-4
Imininingwane:98%min
I-MW:355.43
I-MF:C21H25NO4
Indawo Yokuncibilika:140-1°C
Izinga lokushisa lesitoreji:I-Hygroscopic, Isiqandisi, ngaphansi komkhathi ongasebenzi
Ukuncibilika:I-Chloroform (Kancane), i-Methanol (Kancane)
Umbala:Impuphu Eqinile Emhlophe Kuya Kokungemhlophe


Imininingwane Yomkhiqizo

Amathegi Omkhiqizo

Isingeniso Somkhiqizo

I-Rotundine, eyaziwa nangokuthi i-l-tetrahydropalmatine (l-THP), iyinhlanganisela enezakhiwo zemithi ezithinta uhlelo lwezinzwa oluphakathi kanye nohlelo lwenhliziyo nemithambo yegazi. Kubikwe ukuthi inemiphumela yokudambisa ubuhlungu, yokudambisa, yokukhohlisa, kanye neyokukhathaza. Ngaphezu kwalokho, kuboniswe ukuthi inemiphumela yokuvikela ekulimaleni kobuchopho kanye ne-myocardial ischemia-reperfusion. I-Rotundine yaziwa nangokuthi inamandla okuguqula ukumelana nemithi eminingi kumaseli omdlavuza kanye nezakhiwo zayo zokuvimba iziteshi ze-calcium.
Ingatholakala ezigabeni ze-Stephania tetrandra kanye ne-Corydalis yanhusuo, noma ngezindlela zokwenziwa kwamakhemikhali. Kwenziwe nge-tetrahydropalmatine ngokunciphisa, ukuqhekeka, kanye nokusabela kwe-alkali. I-tetrahydropalmatine ene-iodine ingakhiqizwa nge-tetrahydropalmatine ngokwenziwa kwe-alkali kanye ne-oxidation ukuze kwenziwe okuphindaphindwayo.
Ngokwe-pharmacokinetics, i-Rotundine imuncwa kahle ngemva kokuphathwa ngomlomo futhi isakazwa kakhulu ezicutshini zamafutha, kulandele amaphaphu, isibindi, nezinso. Ikhishwa kakhulu ngezinso. Izifundo kumagundane nonogwaja zikhombisile ukuthi i-Rotundine ingangena emngceleni wegazi nobuchopho futhi ingene ezicutshini zobuchopho, kanti amazinga obuchopho aphansi kunezinga legazi ngemva kwamahora ama-2.
Ngemiphumela emibi, i-Rotundine ingabangela ukozela, isiyezi, ukukhathala, isicanucanu, kanye nokushaqeka ngezinye izikhathi ngenxa yokungezwani komzimba. Izinyathelo zokuphepha zifaka phakathi ukugwema ukusebenzisa kwabesifazane abakhulelwe nabancelisayo, ukuqaphela ukuthi kungenzeka yini ukubekezelela ukusetshenziswa kwesikhathi eside, kanye nokusebenzisa ngokucophelela lapho usebenzisa kanye nama-central nervous system depressants, kanye nokulungiswa okufanele komthamo uma kudingeka.
Ngamafuphi, i-Rotundine iyinhlanganisela enemiphumela eyahlukahlukene yezokwelapha, futhi izakhiwo zayo ziyenza ibe yindaba ethakazelisayo ocwaningweni oluhlukahlukene, okuhlanganisa ukuphathwa kobuhlungu, impilo yenhliziyo, kanye nokwelashwa komdlavuza. Ukuze uthole ulwazi olwengeziwe xhumana nathi.grace@biowaycn.com.

Isici

Ukuqeda ubuhlungu:I-Rotundine iboniswe ukuthi inezakhiwo zokunciphisa ubuhlungu, okwenza iphumelele ekunciphiseni ubuhlungu nokungakhululeki.
Imiphumela yokulwa nokuvuvukala:I-Rotundine ibonise izakhiwo zokulwa nokuvuvukala, ezingasiza ekunciphiseni ukuvuvukala kanye nezimpawu ezihlobene nakho.
Ukuphumula kanye nokudambisa:I-Rotundine isetshenziswe ukukhuthaza ukuphumula nokuzola, okwenza kube wusizo ekulawuleni ukucindezeleka nokukhathazeka.
Umsebenzi we-Antioxidant:Kutholakale ukuthi i-Rotundine ibonisa imiphumela yokulwa nama-antioxidant, engasiza ekuvikeleni amaseli ekulimaleni okubangelwa ama-free radicals.
Kungenzeka ukwelashwa ngokuba umlutha:Ucwaningo oluthile lubonisa ukuthi i-Rotundine ingaba namandla okuphatha umlutha kanye nezimpawu zokuhoxa, ikakhulukazi kulabo abathembele kuma-opioid.
Izinzuzo zesisu:I-Rotundine iye yacwaningwa ngenxa yamandla ayo okunciphisa izinkinga zesisu, njengokuqaqamba kwemisipha kanye nokungakhululeki.

Imininingwane

Ukuhlaziywa Imininingwane
Ukuhlolwa I-Tetrahydropalmatine ≥98%
Ukubukeka Impuphu ephuzi kancane kuya kokumhlophe
Umlotha ≤0.5%
Umswakama ≤5.0%
Izibulala-zinambuzane Okubi
Izinsimbi ezisindayo ≤10ppm
Pb ≤2.0ppm
As ≤2.0ppm
Iphunga Isici
Usayizi wezinhlayiya I-mesh engu-100% kuya ku-80
Izinto eziphilayo:  
Inani lamagciwane ≤1000cfu/g
Isikhunta ≤100cfu/g
I-Salmgosella Okubi
I-Coli Okubi

 

Isicelo

I-Rotundine inezinhlelo zokusebenza ezimbonini eziningana, okuhlanganisa:
Imboni Yezemithi:I-Rotundine isetshenziswa embonini yezemithi ngenxa yezakhiwo zayo ezingaba yisidambisi-zinhlungu, isilalisi, kanye ne-anxiolytic. Ingafakwa emithini yokulawula ubuhlungu kanye nokuqeda ukukhathazeka.
Ukunakekelwa Kwempilo Nokuphila Kahle:Ngenxa yezinzuzo zayo zezempilo ezibikiwe, i-Rotundine ingasetshenziswa emikhiqizweni yezempilo kanye nenhlalakahle ehlose ukukhuthaza ukuphumula nokulawula ubuhlungu.
Ucwaningo Nentuthuko:I-Rotundine inentshisekelo emizamweni yocwaningo nentuthuko egxile empilweni yenhliziyo nemithambo yegazi, ukwelashwa komdlavuza, kanye nezimo zezinzwa ngenxa yemiphumela yayo ebikiwe kulezi zinhlelo.
Izakhamzimba:Kukhona amathuba okufakwa kwe-Rotundine emikhiqizweni ye-nutraceutical eyenzelwe ukusekela impilo kanye nenhlalakahle iyonke.
Kubalulekile ukuqaphela ukuthi ukusetshenziswa kwe-Rotundine kungahluka ngokuya ngokuvunyelwa kwemithetho kanye nocwaningo oluqhubekayo embonini ngayinye.

Imininingwane Yokukhiqiza

Imikhiqizo yethu ikhiqizwa kusetshenziswa izindlela zokulawula ikhwalithi eziqinile futhi ilandela amazinga aphezulu ezinqubo zokukhiqiza. Sibeka phambili ukuphepha nekhwalithi yomkhiqizo wethu, siqinisekisa ukuthi uhlangabezana nezidingo zomthetho kanye nezitifiketi zemboni. Lokhu kuzibophezela kwikhwalithi kuhlose ukwakha ukwethembana nokuqiniseka ekuthembekeni komkhiqizo wethu. Inqubo yokukhiqiza ejwayelekile imi kanje:

Ukupakishwa kanye Nesevisi

Isitoreji:Gcina endaweni epholile, eyomile, nehlanzekile, Vikela emswakama nasekukhanyeni okuqondile.
Iphakheji Eningi:20~25kg/isigubhu.
Isikhathi esiholayo:Izinsuku eziyi-7 ngemuva kwe-oda lakho.
Isikhathi Sokuphila Seshelufu:iminyaka engu-2.
Phawula:Imininingwane eyenziwe ngokwezifiso ingafinyelelwa.

Izindlela Zokukhokha Nokulethwa

I-Express
Ngaphansi kwe-100kg, izinsuku ezi-3-5
Isevisi yokungena emnyango kulula ukuyithatha izimpahla

Ngasolwandle
Ngaphezulu kwama-300kg, cishe izinsuku ezingama-30
Kudingeka umthengisi wezinsizakalo zokukhishwa kwemvume ochwepheshe

Ngomoya
100kg-1000kg, Izinsuku ezi-5-7
Kudingeka umthengisi wezinsizakalo zokuhlanza ochwepheshe kusukela esikhumulweni sezindiza kuya esikhumulweni sezindiza

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Isitifiketi

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